Stefan Knapp
机构: University of Frankfurt
每年引用次数
引用次数
引用: 48,112
H-指数: 112
I10-指数 : 391
出版物: 723
On the stability of proteins from hyperthermophiles : A structural and thermodynamic study
Stefan Knapp
1996
The global cancer genomics consortium's symposium: new era of molecular medicine and epigenetic cancer medicine - cross section of genomics and epigenetics
Rajendra Badwe , Stefan Knapp , M. Radhakrishna Pillai , Luis Costa
Genes & Cancer 6 1 -8
2015
Development of SRPK1 inhibitors as novel anti-angiogenic therapeutics for exudative age-related macular degeneration (AMD)
Roya Babaei-Jadidi , Stephen Wearmouth , Hamish Troop , Jonathan Rowlinson
Investigative Ophthalmology & Visual Science 56 ( 7) 2461 -2461
2015
The global cancer genomics consortium’s third annual symposium: From oncogenomics to cancer care
Stefan Knapp , Sandra Casimiro , Masakazu Toi , Maria Carmo-Fonseca
Genes & Cancer 5 64 -70
2
2014
Discovery of novel inhibitors of the phosphatase activity of the soluble epoxide hydrolase
Ewgenij Proschak , Denys Pogoryelov , G. Enrico Rovati , Dieter Steinhilber
The FASEB Journal 32
1
2018
Integrated analysis of Shank1 PDZ interactions with C-terminal and internal binding motifs
Muhammad Ali , Mishal Mariam McAuley , Susanne Lüchow , Stefan Knapp
Current Research in Structural Biology 3 41 -50
2021
Structure-kinetic relationship reveals the mechanism of selectivity of FAK inhibitors over PYK2.
Ariane Nunes-Alves , Iva Navratilova , Daria B. Kokh , Stefan Knapp
Chemistry & Biology 28 ( 5)
2021
Drugging the “Undruggable” MYCN Oncogenic Transcription Factor: Overcoming Previous Obstacles to Impact Childhood Cancers
Kevan M. Shokat , Yaël P. Mossé , Yaël P. Mossé , Steven J. Metallo
Cancer Research 81 ( 7) 1627 -1632
2021
Deciphering the LRRK code: LRRK1 and LRRK2 phosphorylate distinct Rab proteins and are regulated by diverse mechanisms.
Dario R Alessi , Sebastian Mathea , Stefan Knapp , Robert Gourlay
Biochemical Journal 478 ( 3) 553 -578
2021
Development of a potent and selective chemical probe for the pleiotropic kinase CK2.
Laszlo Gyenis , David W. Litchfield , Stefan Knapp , Stefan Knapp
Chemistry & Biology 28 ( 4)
34
2021
Combined Cardioprotective and Adipocyte Browning Effects Promoted by the Eutomer of Dual sEH/PPARγ Modulator.
Ewgenij Proschak , Ewgenij Proschak , Pamela Fischer-Posovszky , Lilia Weizel
Journal of Medicinal Chemistry 64 ( 5) 2815 -2828
2021
Highly selective inhibitors of protein kinases CLK and HIPK with the furo[3,2-b]pyridine core.
Kamil Paruch , Apirat Chaikuad , Karel Souček , Stefan Knapp
European Journal of Medicinal Chemistry 215 113299
2021
Demonstrating Ligandability of the LC3A and LC3B Adapter Interface
Volker Dötsch , Ewgenij Proschak , Ewgenij Proschak , Dalibor Odadzic
Journal of Medicinal Chemistry 64 ( 7) 3720 -3746
2021
Structure and Inhibitor Binding Characterization of Oncogenic MLLT1 Mutants.
Apirat Chaikuad , Apirat Chaikuad , Stefan Knapp , Stefan Knapp
ACS Chemical Biology 16 ( 4) 571 -578
2021
7-(2-Anilinopyrimidin-4-yl)-1-benzazepin-2-ones Designed by a “Cut and Glue” Strategy Are Dual Aurora A/VEGF-R Kinase Inhibitors
Conrad Kunick , Apirat Chaikuad , Apirat Chaikuad , Frank Totzke
Molecules 26 ( 6) 1611
2021
Structural Insights into Plasticity and Discovery of Remdesivir Metabolite GS-441524 Binding in SARS-CoV-2 Macrodomain
Xiaomin Ni , Martin Schröder , Vincent Olieric , May E Sharpe
ACS Medicinal Chemistry Letters 12 ( 4) 603 -609
2
2021
Oxaprozin Analogues as Selective RXR Agonists with Superior Properties and Pharmacokinetics.
Ewgenij Proschak , Apirat Chaikuad , Apirat Chaikuad , Daniel Merk
Journal of Medicinal Chemistry 64 ( 8) 5123 -5136
7
2021
Exploiting vulnerabilities of SWI/SNF chromatin remodelling complexes for cancer therapy.
Andreas C Joerger , Andreas C Joerger , Stefan Knapp , Marek Wanior
Oncogene 40 ( 21) 3637 -3654
2021
Endogenous vitamin E metabolites mediate allosteric PPARγ activation with unprecedented co-regulatory interactions
Oliver Werz , Manfred Schubert-Zsilavecz , Apirat Chaikuad , Daniel Merk
Chemistry & Biology
14
2021
A Chemical Toolbox for Labeling and Degrading Engineered Cas Proteins
Jie Chen , Stefan Knapp , Guangqi Song , Xinlai Cheng
JACS Au
2021
Panagis Filippakopoulos Oleg Fedorov Apirat Chaikuad Paul E Brennan Frank von Delft Brian Marsden Wen Hwa Lee Cheryl Arrowsmith Sebastian Mathea Benjamin E. Turk Jeyanthy Eswaran Chas Bountra Opher Gileadi Martin Schröder Juerg Schwaller Ashley Pike Kilian V. M. Huber Stuart J Conway James Bradner Laurent Meijer