In search for the active metabolites and the cellular target of the antitubercular prodrug TP053

M Manfredi , L Chiarelli , Makarov , E Marengo
Tuberculosis Drug Discovery & Development Gordon Research Conference 25-30/06

2017
Identification and characterization of the cellular target for benzothiazinones, a new potential antitubercular drug class.

Giulia Manina , V Makarov , MARIA ROSALIA Pasca , O Ryabova
Congrex Sweden AB 3 -3

1
2008
Rv3790 is the cellular target for benzothiazinones, a new promising antitubercular drug class

Giulia Manina , V Makarov , MARIA ROSALIA Pasca , O Ryabova
Azuleon meetings 10 D02 -D04

2008
Isolation of mycobacterial monooxygenase EthA

M Zahorszka , J Madacki , D Mikulasova , J Kordulakova
FEBS OPEN BIO 8 418 -419

2018
Investigation of the effect of tuberculosis drug isoxyl on selected mycobacterial epoxide hydrolases

J Madacki , M Kopal , M Jackson , J Kordulakova
FEBS JOURNAL 280 355 -356

2013
Biochemical characterization of acyltransferase MSMEG_2934 from Mycobacterium smegmatis

Z Svetlikova , J Kordulakova , K Mikusova ,
FEBS JOURNAL 280 361 -361

2013
Identification of a Novel Galactosyl Transferase Involved in Biosynthesis of the Mycobacterial Cell Wall

Katarína Mikušová , Martina Beláňová , Jana Korduláková , Kristine Honda
Journal of Bacteriology 188 ( 18) 6592 -6598

59
2006
Isoxyl Activation Is Required for Bacteriostatic Activity against Mycobacterium tuberculosis

Jana Korduláková , Yves L. Janin , Avraham Liav , Nathalie Barilone
Antimicrobial Agents and Chemotherapy 51 ( 11) 3824 -3829

29
2007
Trehalose Conjugation Enhances Toxicity of Photosensitizers against Mycobacteria.

Amit K Dutta , Eira Choudhary , Xuan Wang , Monika Záhorszka
ACS central science 5 ( 4) 644 -650

5
2019
Investigation of ABC transporter from mycobacterial arabinogalactan biosynthetic cluster.

P. Dianišková , J. Korduláková , H. Škovierová , D. Kaur
General Physiology and Biophysics 30 ( 3) 239 -250

15
2011
A Coumarin-Based Analogue of Thiacetazone as Dual Covalent Inhibitor and Potential Fluorescent Label of HadA in Mycobacterium tuberculosis.

Jana Korduláková , Stefan Chassaing , Stefan Chassaing , Maria Rosalia Pasca
ACS Infectious Diseases 7 ( 3) 552 -565

2021
Mycobacterial Epoxide Hydrolase EphD Is Inhibited by Urea and Thiourea Derivatives

Jana Korduláková , Jan Madacki , Martin Kopál , Mary Jackson
International Journal of Molecular Sciences 22 ( 6) 2884

2021
An ABC transporter Wzm-Wzt catalyzes translocation of lipid-linked galactan across the plasma membrane in mycobacteria.

Stanislav Kozmon , Katarína Mikušová , Michal Kaliňák , Jana Korduláková
Proceedings of the National Academy of Sciences of the United States of America 118 ( 17)

2
2021
Genetic Basis for the Biosynthesis of Methylglucose Lipopolysaccharides inMycobacterium tuberculosis

Gustavo Stadthagen , Tounkang Sambou , Marcelo Guerin , Nathalie Barilone
Journal of Biological Chemistry 282 ( 37) 27270 -27276

50
2007
7
2014
Covalent modification of the Mycobacterium tuberculosis FAS-II dehydratase by Isoxyl and Thiacetazone.

Anna E. Grzegorzewicz , Nathalie Eynard , Annaïk Quémard , E. Jeffrey North
ACS Infectious Diseases 1 ( 2) 91 -97

29
2015