The orphan receptor GPR55 is a novel cannabinoid receptor. Commentary
R. G. Pertwee , S. Hjorth , J. Leonova , T. Drmota
British Journal of Pharmacology 152 ( 7)
7
2007
Diversity in the signalling and regulation of G-protein-coupled receptors.
G. Milligan , D. A. Groarke , A. McLean , R. Ward
Biochemical Society Transactions 27 ( 2) 149 -154
6
1999
Visualising signal initiation and termination by G protein-coupled receptors
G. Milligan , T. Drmota , D. S. Bahia , D. A. Groarke
Biochemical Society Transactions 28 ( 5)
2000
SAT0245 Azd9567: a novel oral selective glucocorticoid receptor modulator, demonstrated to have an improved therapeutic ratio compared to prednisolone in pre-clinical studies, is safe and well tolerated in first clinical study.
R. Hendrickx , T. Hegelund-Myrbäck , M. Dearman , S. Prothon
Annals of the Rheumatic Diseases 77 984 -985
1
2018
Adenosine is not a direct GHSR agonist--artificial cross-talk between GHSR and adenosine receptor pathways.
N.-O. Hermansson , D. G. A. Morgan , T. Drmota , N. Larsson
Acta Physiologica 190 ( 1) 77 -86
9
2007
Occurrence and pharmacological characterization of four human tachykinin NK2 receptor variants
Ingela Ahlstedt , Susanna Engberg , John Smith , Chris Perrey
Biochemical Pharmacology 76 ( 4) 476 -481
4
2008
Molecular cloning, mutations and effects of NK1 receptor antagonists reveal the human-like pharmacology of gerbil NK1 receptors
Susanna Engberg , Ingela Ahlstedt , Agnes Leffler , Erik Lindström
Biochemical Pharmacology 73 ( 2) 259 -269
16
2007
Senktide-induced gerbil foot tapping behaviour is blocked by selective tachykinin NK1 and NK3 receptor antagonists
Elin Kristensson , Rebecka Adolfsson , Agnes Leffler , Ingela Ahlstedt
European Journal of Pharmacology 577 ( 1) 78 -86
9
2007
Discovery of a Novel Oral Glucocorticoid Receptor Modulator (AZD9567) with Improved Side Effect Profile.
Lena Ripa , Karl Edman , Matthew Dearman , Goran Edenro
Journal of Medicinal Chemistry 61 ( 5) 1785 -1799
49
2018
Discovery of AZD6642, an inhibitor of 5-lipoxygenase activating protein (FLAP) for the treatment of inflammatory diseases.
Malin Lemurell , Johan Ulander , Susanne Winiwarter , Anders Dahlén
Journal of Medicinal Chemistry 58 ( 2) 897 -911
28
2015
Diversity in the signaling and regulation of G protein-coupled receptors
Graeme Milligan , D. Alex. Groake , Alison MacLean , Richard Ward
Biochemical Society Transactions 27 ( 1)
1
1999
Design of small molecule inhibitors of acetyl-CoA carboxylase 1 and 2 showing reduction of hepatic malonyl-CoA levels in vivo in obese Zucker rats.
Christoffer Bengtsson , Stefan Blaho , David Blomberg Saitton , Kay Brickmann
Bioorganic & Medicinal Chemistry 19 ( 10) 3039 -3053
30
2011
Inhibition of AMP Deaminase Activity Does Not Improve Glucose Control in Rodent Models of Insulin Resistance or Diabetes
Therese Admyre , Lena Amrot-Fors , Maria Andersson , Martin Bauer
Chemistry & Biology 21 ( 11) 1486 -1496
11
2014
Agonist-induced Internalization of the G Protein G11α and Thyrotropin-releasing Hormone Receptors Proceed on Different Time Scales
Tomas Drmota , Jiri Novotny , Gun-Do Kim , Karin A. Eidne
Journal of Biological Chemistry 273 ( 34) 21699 -21707
41
1998
Real Time Visualization of Agonist-mediated Redistribution and Internalization of a Green Fluorescent Protein-tagged Form of the Thyrotropin-releasing Hormone Receptor
Tomas Drmota , Gwyn W. Gould , Graeme Milligan
Journal of Biological Chemistry 273 ( 37) 24000 -24008
54
1998
Functional analysis of a human A1 adenosine receptor/green fluorescent protein/Gi1α fusion protein following stable expression in CHO cells
Nicola Bevan , Tim Palmer , Tomas Drmota , Alan Wise
FEBS Letters 462 ( 1) 61 -65
19
1999
Analysis of the C-terminal tail of the rat thyrotropin-releasing hormone receptor-1 in interactions and cointernalization with β-arrestin 1-green fluorescent protein
D Alex Groarke , Tomas Drmota , Daljit S Bahia , Nicholas A Evans
Molecular Pharmacology 59 ( 2) 375 -385
57
2001
CELL BIOLOGY AND METABOLISM-Real time visualization of agonist-mediated redistribution and internalization of a green fluorescent protein-tagged form of the thyrotropin-releasing hormone receptor
Tomas Drmota , Gwyn W Gould , Graeme Milligan
Journal of Biological Chemistry 273 ( 37) 24000 -24008
1998
From lead to candidate drug selection of AZD6642, a 5-lipoxygenase activating protein (FLAP) inhibitor
Malin Lemurell , Jonas Barlind , Johan Broddefalk , Anders Dahlen
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 247
2014
The discovery of a selective and potent A2a agonist with extended lung retention
Annika BM Åstrand , Eva Lamm Bergström , Hui Zhang , Lena Börjesson
Pharmacology Research & Perspectives 3 ( 3) e00134 -e00134
10
2015