Novel antimicrobial strategies to treat multi‐drug resistant Staphylococcus aureus infections

Edward JA Douglas , Sri W Wulandari , Scott D Lovell , Maisem Laabei
Microbial biotechnology 16 ( 7) 1456 -1474

12
2023
A Suite of Activity-Based Probes To Dissect the KLK Activome in Drug-Resistant Prostate Cancer.

Charlotte L Bevan , Thomas Kryza , Judith A Clements , Edward W Tate
Journal of the American Chemical Society

2021
Substrate-biased activity-based probes identify proteases that cleave receptor CDCP1.

Sean Porazinski , Sean Porazinski , Hannu Koistinen , Marina Pajic
Nature Chemical Biology 1 -8

14
2021
Depsipeptides Featuring a Neutral P1 Are Potent Inhibitors of Kallikrein-Related Peptidase 6 with On-Target Cellular Activity

Elena De Vita , Peter Schüler , Scott Lovell , Jasmin Lohbeck
Journal of Medicinal Chemistry 61 ( 19) 8859 -8874

11
2018
Targeting STAT3 signaling using stabilised sulforaphane (SFX-01) inhibits endocrine resistant stem-like cells in ER-positive breast cancer

Bruno M. Simões , Angélica Santiago-Gómez , Chiara Chiodo , Tiago Moreira
Oncogene 39 ( 25) 4896 -4908

2020
Challenges for targeting SARS-CoV-2 proteases as a therapeutic strategy for COVID-19

Kas Steuten , Heeyoung Kim , John C. Widen , Brett M. Babin
bioRxiv

56
2020
Identification of highly selective covalent inhibitors by phage display.

Shiyu Chen , Scott Lovell , Sumin Lee , Matthias Fellner
Nature Biotechnology 39 ( 4) 490 -498

37
2021
The molecular function of kallikrein-related peptidase 14 demonstrates a key modulatory role in advanced prostate cancer

Thomas Kryza , Nathalie Bock , Scott Lovell , Anja Rockstroh
Molecular Oncology 14 ( 1) 105 -128

4
2020
Strategies for Tuning the Selectivity of Chemical Probes that Target Serine Hydrolases

Franco Faucher , John M. Bennett , Matthew Bogyo , Scott Lovell
Chemistry & Biology 27 ( 8) 937 -952

8
2020
Novel and versatile synthesis of disubstituted 1,2-dihydro-1,2,4-triazol-3-ones.

Mark A. Graham , Paul A. Bethel , Jonathan Burgess , Gary Fairley
Organic Letters 15 ( 23) 6078 -6081

5
2013
Faecal neutrophil elastase-antiprotease balance reflects colitis severity.

Rachael Barry , David Ruano-Gallego , Shiva T Radhakrishnan , Scott Lovell
Mucosal Immunology 13 ( 2) 322 -333

11
2020
Chemical Probes for Proteins and Networks

Scott Lovell , Charlotte L. Sutherell , Edward W. Tate
Mass Spectrometry‐Based Chemical Proteomics 127 -158

2019
A KLK6 activity-based probe reveals a role for KLK6 activity in pancreatic cancer cell invasion

Leran Zhang , Scott Lovell , Elena De Vita , Pravin Kumar Ankush Jagtap
Journal of the American Chemical Society 144 ( 49) 22493 -22504

8
2022
Solid phase synthesis of fluorosulfate containing macrocycles for chemoproteomic workflows

Franco F Faucher , Daniel Abegg , Phillip Ipock , Alexander Adibekian
Israel Journal of Chemistry 63 ( 3-4) e202300020 -e202300020

4
2023
Mixed alkyl/aryl phosphonates identify metabolic serine hydrolases as antimalarial targets

John M Bennett , Sunil K Narwal , Stephanie Kabeche , Daniel Abegg
Cell Chemical Biology

2024