Rapid microwave-assisted Suzuki coupling on solid-phase
作者： Mats Larhed , Gunnar Lindeberg , Anders Hallberg
DOI: 10.1016/0040-4039(96)01872-2
关键词: Chemistry 、 Phase (matter) 、 Suzuki reaction 、 Combinatorial chemistry 、 Aryl 、 Microwave assisted 、 Organic chemistry 、 TentaGel-S
摘要: Abstract Microwave-assisted palladium-catalysed coupling of aryl and heteroaryl boronic acids with iodo- bromo-substituted benzoic acids, anchored to TentaGel S RAM, provided high isolated yields coupled products after a reaction time 3.8 minutes (45 W).
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