Synthesis of imidazo[1,2-a]pyridines: a decade update

作者: Avik Kumar Bagdi , Sougata Santra , Kamarul Monir , Alakananda Hajra

DOI: 10.1039/C4CC08495K

关键词: Bicyclic moleculeOxidative coupling of methaneOrganic chemistryCombinatorial chemistryImidazopyridineScaffoldHydroaminationMoietyChemistry

摘要: Imidazopyridine is one of the important fused bicyclic 5–6 heterocycles and it recognized as a “drug prejudice” scaffold due to its wide range applications in medicinal chemistry. This moiety also useful material science because structural character. Synthesis this from easily available chemicals desirable tremendous use various branches Here we report review on synthesis employing different strategies such condensation, multicomponent reactions, oxidative coupling, tandem aminooxygenation, hydroamination reactions.

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