Compounds useful for treating diseases caused by retroviruses

作者: Didier Scherrer , Romain Najman , Noëlie Campos , Aude Garcel , Jamal Tazi

DOI:

关键词: AlkylPyrimidineStereochemistryPyrazineHalogenGroup (periodic table)Pyridazine2-groupChemistryAlkoxy group

摘要: Methods for preventing or treating retroviral infection not HIV and/or preventing, inhibiting a disease caused by the include contacting cell with compound (I) wherein: means pyridazine, pyrimidine pyrazine group, R independently represent hydrogen atom, halogen atom group chosen among —CN, hydroxyl, —COOR 1 , (C -C 3 )fluoroalkyl, )fluoroalkoxy, —NO 2 —NR 4 )alkoxy, phenoxy and )alkyl alkyl being optionally mono-substituted hydroxyl n is 1, 3, n′ 2, R′ morpholinyl morpholino N-methylpiperazinyl )fluoroalkyl )alkoxy —CN Z N C, Y X W T U C.

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