Synthesis and antibacterial activity of emodin and its derivatives against methicillin-resistant Staphylococcus aureus
作者： Thidarat Chalothorn , Vatcharin Rukachaisirikul , Souwalak Phongpaichit , Sakawrat Pannara , Chittreeya Tansakul
DOI: 10.1016/J.TETLET.2019.151004
关键词: Medicinal chemistry 、 Vero cell 、 Cytotoxicity 、 Acylation 、 Ammonium 、 Chemistry 、 Methyl group 、 Emodin 、 Staphylococcus aureus 、 Antibacterial activity 、 Organic chemistry 、 Biochemistry 、 Drug discovery
摘要: … Synthesis of the antibacterial emodin was improved using Friedel-Crafts acylation as a key step leading to 37% overall yield. In addition, 21 analogues were synthesized by structural …
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