4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide
作者： Alexander Flohr , Sonia Maria Poli , Claus Riemer , Jean-Luc Moreau , Lucinda Steward
DOI:
关键词: Substance abuse 、 Ethanol 、 Amide 、 Carboxylic acid 、 Neuroprotection 、 Medicine 、 Drug 、 Nicotine 、 Piperidine 、 Pharmacology
摘要: The present invention relates to the compound of formula (I): which is 4-hydroxy-4-methyl-piperidine-l-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide, and pharmaceutically acceptable addition salts thereof. It has been found that useful for treatment or prevention Alzheimer's disease, Parkinson's Huntington's neuroprotection, schizophrenia, anxiety, pain, respiration deficits, depression, ADHD ( attention deficit hyper-activity disorder), drug addiction amphetamines, cocaine, opioids, ethanol, nicotine, cannabinoids, asthma, allergic responses, hypoxia, ischemia, seizure, substance abuse, use as muscle relaxants, antipsychotics, antiepileptics, anticonvulsants cardioprotective agents.
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