Benzimidazole anthelmintic agents.
作者： Alexander Crossan Goudie , Christopher James Dutton , Bernard Joseph Pfizer Ce Banks
DOI:
关键词: Anthelmintic 、 Alkyl 、 Benzimidazole 、 Medicinal chemistry 、 Chemistry
摘要: Benzimidazole anthelmintic agents of formula (I) and their non-toxic salts in which R is H, CO2(C1-C10 alkyl), -CO2(cholester-3-yl) or -CO2(CH2)COOH -CO2(CH2)nCO2(C1-C6 n = 1 to 10, R1 optionally substituted benzoyl, phenyloxy, phenylthio, phenylsulfonyl, phenylsulfinyl, phenylsulfonyloxy, alkylthio, alkylsulfinyl, alkylsulfonyl, cycloalkylcarbonyl selected from a variety heterocyclic groups R?2 R3? are independently -CO?2?(C1-C4 alkyl).
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