Direct solid-phase synthesis of quinoxaline-containing peptides
作者： Anna Staszewska , Piotr Stefanowicz , Zbigniew Szewczuk
DOI: 10.1016/J.TETLET.2005.06.047
关键词: Quinoxaline 、 Chemistry 、 Solid-phase synthesis 、 Alanine 、 Residue (chemistry) 、 Organic chemistry
摘要: The solid-phase synthesis of a series model dipeptides containing various 3-(quinoxalin-6-yl)alanine analogues is described. method involves formation quinoxaline heterocycle by condensation between an α-dicarbonyl compound and β-(3,4-diaminophenyl)alanine residue, immobilized on solid support.
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