Indolylboronic Acids: Preparation and Applications

作者: Marek Čubiňák , Tereza Edlová , Peter Polák , Tomáš Tobrman

DOI: 10.3390/MOLECULES24193523

关键词: ElectrophileSuzuki reactionBoronic acidCombinatorial chemistryChemistryIndole testMaterial chemistry

摘要: Indole derivatives are associated with a variety of both biological activities and applications in the field material chemistry. A number different strategies for synthesizing substituted indoles by means reactions indolylboronic acids electrophilic compounds considered methods choice modifying because easily available, stable, non-toxic new using have been described literature. Thus, aim this review is to summarize available preparation as well their chemical transformations. The covers period 2010–2019.

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