Bicyclic heterocycles, the preparation thereof, and their use as pharmaceuticals
作者： Norbert Hauel , Henning Priepke , Jean-Marie Stassen , Uwe Ries , Wolfgang Weinen
DOI:
关键词: Stereochemistry 、 Bicyclic molecule 、 Group (periodic table) 、 Tautomer 、 Chemistry
摘要: The present invention relates to 5-membered heterocyclic condensed benzoderivatives of formula ##STR1## wherein Ra Rc, A, X and Y are defined as in claim 1, the tautomers, stereoisomers, mixtures thereof salts thereof, particularly physiologically acceptable with inorganic or organic acids bases which have valuable properties. compounds above I Rc denotes a cyano group intermediates for preparing other I, one following amidino groups tautomers stereoisomers pharmacological properties, an antithrombotic activity.
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