New benzamide derivatives as bradykinin antagonists
作者： Monika Vastag , Sandor Farkas , Gyorgy Keseru , Eva Schmidt , Istvan Vago
DOI:
关键词: Bradykinin 、 Benzamide 、 Stereochemistry 、 Chemistry
摘要: The present invention relates to new phenylsulfamoyl benzamide derivatives of formula (I), wherein R1-R5 and Z are as defined in the claims, optical antipodes or racemates and/or salts hydrates solvates thereof, which selective antagonists bradykinin B1, processes for producing these compounds, pharmacological compositions containing them their use therapy prevention painful inflammatory conditions.
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