Cyclized peptidomimetic small molecule inhibitors of the wdr5 and mll1 interaction
作者： Hacer Karatas , Denzil Bernard , Yali Dou , Fang Cao , Shaomeng Wang
DOI:
关键词: Stereochemistry 、 Combinatorial chemistry 、 Chemistry 、 Small molecule 、 Peptidomimetic 、 WDR5
摘要: Cyclic peptidomimetics that inhibit the interaction between MLL1 and WDR5 are disclosed. Methods of inhibiting activity methods treating cancers also
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