Forecasting the oral absorption behavior of poorly soluble weak bases using solubility and dissolution studies in biorelevant media.
作者： Edmund S. Kostewicz , Ulrich Brauns , Robert Becker , Jennifer B. Dressman
关键词: Pharmacology toxicology 、 Chemical engineering 、 Organic chemistry 、 Weak base 、 Solubility 、 Dissolution 、 Absorption (chemistry) 、 Chemistry
摘要:
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sci-hub.se 参考文章(13)
Eleftheria Nicolaides, Eric Galia, Constantin Efthymiopoulos, Jennifer B. Dressman, Christos Reppas, Forecasting the In Vivo Performance of Four Low Solubility Drugs from Their In Vitro Dissolution Data Pharmaceutical Research. ,vol. 16, pp. 1876- 1882 ,(1999) , 10.1023/A:1018959511323
E. Galia, E. Nicolaides, D. Hörter, R. Löbenberg, C. Reppas, J. B. Dressman, Evaluation of Various Dissolution Media for Predicting In Vivo Performance of Class I and II Drugs Pharmaceutical Research. ,vol. 15, pp. 698- 705 ,(1998) , 10.1023/A:1011910801212
Jennifer B. Dressman, Rosemary R. Berardi, Lambros C. Dermentzoglou, Tanya L. Russell, Stephen P. Schmaltz, Jeffrey L. Barnett, Kathleen M. Jarvenpaa, Upper gastrointestinal (GI) pH in young, healthy men and women. Pharmaceutical Research. ,vol. 7, pp. 756- 761 ,(1990) , 10.1023/A:1015827908309
Jennifer B. Dressman, Gordon L. Amidon, Christos Reppas, Vinod P. Shah, Dissolution Testing as a Prognostic Tool for Oral Drug Absorption: Immediate Release Dosage Forms Pharmaceutical Research. ,vol. 15, pp. 11- 22 ,(1998) , 10.1023/A:1011984216775
Tanya L. Russell, Rosemary R. Berardi, Jeffrey L. Barnett, Tami L. O’Sullivan, John G. Wagner, Jennifer B. Dressman, pH-Related Changes in the Absorption of Dipyridamole in the Elderly Pharmaceutical Research. ,vol. 11, pp. 136- 143 ,(1994) , 10.1023/A:1018918316253
Theodore R. Bates, Milo Gibaldi, Joseph L. Kanig, Solubilizing Properties of Bile Salt Solutions II. Journal of Pharmaceutical Sciences. ,vol. 55, pp. 901- 906 ,(1966) , 10.1002/JPS.2600550906
Arne Melander, Influence of Food on the Bioavailability of Drugs Clinical Pharmacokinectics. ,vol. 3, pp. 337- 351 ,(1978) , 10.2165/00003088-197803050-00001
Theodore R. Bates, Milo Gibaldi, Joseph L. Kanig, Solubilizing Properties of Bile Salt Solutions I Journal of Pharmaceutical Sciences. ,vol. 55, pp. 191- 199 ,(1966) , 10.1002/JPS.2600550213
L. Ovesen, F. Bendtsen, U. Tage-Jensen, N.T. Pedersen, B.R. Gram, S.J. Rune, Intraluminal pH in the stomach, duodenum, and proximal jejunum in normal subjects and patients with exocrine pancreatic insufficiency Gastroenterology. ,vol. 90, pp. 958- 962 ,(1986) , 10.1016/0016-5085(86)90873-5
Terhaag B, Feller K, Donath F, Le Petit G, The absolute and relative bioavailability of dipyridamole from different preparations and the in vitro-in vivo comparison. International journal of clinical pharmacology, therapy, and toxicology. ,vol. 24, pp. 298- 302 ,(1986)