1,3,4-oxadiazine derivatives and their use as pesticides
作者： Christoph Erdelen , Andrew Plant , Hubert Dyker , Achim Harder , Juergen Scherkenbeck
DOI:
关键词: Aryl 、 Medicinal chemistry 、 Ring (chemistry) 、 Chemistry 、 Alkyl 、 Stereochemistry
摘要: The invention concerns novel (1,3,4)-oxadiazine derivatives of formula (I) in which: R?1 and R2?, independently each other, stand for hydrogen, or alkyl, hydroxylalkyl, alkanoyloxyalkyl, alkoxyalkyl, arylalkoxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, carboxyalkyl, alkoxycarbonylalkyl, aryloxycarbonylalkyl, arylalkyloxycarbonylalkyl, carbamoylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkoxycarbonylaminoalkyl, alkylcarbonyl, cycloalkylcarbonyl case optionally substituted by halogen, cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, arylcarbonyl, heterocyclylalkyl, hetaryl hetarylalkyl; R1, R2 the two nitrogen atoms to which they are bonded an heterocyclic ring; R?3 R4?, alkenyl, hydroxyalkyl, R4? jointly alkylene group (a), R?5 R6?, alkylcarbonyl Q?1 Q2?, oxygen sulphur, 6,6-diphenyl-(1,3,4)-oxadiazinane-2,5-dione being excluded. also a process preparing these substances their use as pesticides endoparasites.
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