SYNTHESIS OF SOME SACCHARIN DERIVATIVES OF EXPECTED BIOLOGICAL ACTIVITY BASED ON N-(SACCHARINYL)-ACETIC ACID AZIDE
作者： M. M. H. Arief
DOI: 10.1080/10426509608046419
关键词: Acetic acid 、 Catalysis 、 Base (chemistry) 、 Organic chemistry 、 Decomposition 、 Glycine 、 Chloride 、 Chemistry 、 Azide 、 Lewis acids and bases
摘要: Abstract Azide was prepared from the corresponding acid chloride . The base catalyzed decomposition with aromatic amines, aminobenzoic acids and/or hydrazines afforded anilides hydrazides via azido group displacement. Compounds and were refluxed in Ac2O to give 1,3,4-oxadiazole derivatives Lewis of azide anhyd. AlCl3 dry substrates gave ketones Also, reaction glycine
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