Compositions of buprenorphine and μ antagonists

作者: Daniel Deaver , Elliot Ehrich

DOI:

关键词: Activity indexBuprenorphineChemistryOpioid receptorAgonist-antagonistPharmacologyAntagonist

摘要: The invention relates to a composition comprising buprenorphine and μ opioid receptor antagonist, wherein the is characterized by an Agonist Antagonist Activity Index (AAnAI) of between about 0.7 2.2; wherein;

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