Farmaci interferenti sull’azione recettoriale dei glicocorticoidi

Kimmo Kontula, Timo Paavonen, Tapani Luukkainen, Leif C. Andersson, Binding of progestins to the glucocorticoid receptor Biochemical Pharmacology. ,vol. 32, pp. 1511- 1518 ,(1983) , 10.1016/0006-2952(83)90474-4

Richard Poulin, Denis Baker, Donald Poirier, Fernand Labrie, Multiple actions of synthetic ‘progestins’ on the growth of ZR-75-1 human breast cancer cells: Anin vitro model for the simultaneous assay of androgen, progestin, estrogen, and glucocorticoid agonistic and antagonistic activities of steroids Breast Cancer Research and Treatment. ,vol. 17, pp. 197- 210 ,(1991) , 10.1007/BF01806369

XAVIER BERTAGNA, CHRISTINE BERTAGNA, JEAN-PIERRE LUTON, JEAN-MARC HUSSON, FRANÇOIS GIRARD, The new steroid analog RU 486 inhibits glucocorticoid action in man. The Journal of Clinical Endocrinology and Metabolism. ,vol. 59, pp. 25- 28 ,(1984) , 10.1210/JCEM-59-1-25

R. C. Gaillard, A. Riondel, A. F. Muller, W. Herrmann, E. E. Baulieu, RU 486: a steroid with antiglucocorticosteroid activity that only disinhibits the human pituitary-adrenal system at a specific time of day Proceedings of the National Academy of Sciences of the United States of America. ,vol. 81, pp. 3879- 3882 ,(1984) , 10.1073/PNAS.81.12.3879

Patrick Poyet, Fernand Labrie, Comparison of the antiandrogenic/androgenic activities of flutamide, cyproterone acetate and megestrol acetate. Molecular and Cellular Endocrinology. ,vol. 42, pp. 283- 288 ,(1985) , 10.1016/0303-7207(85)90059-0

Marianne Mann, Glucocorticoidlike Activity of Megestrol: A Summary of Food and Drug Administration Experience and a Review of the Literature JAMA Internal Medicine. ,vol. 157, pp. 1651- 1656 ,(1997) , 10.1001/ARCHINTE.1997.00440360053005

Oskari Heikinheimo, Taneli Raivio, Helena Honkanen, Sirpa Ranta, Olli A. Jänne, Termination of Pregnancy with Mifepristone and Prostaglandin Suppresses Transiently Circulating Glucocorticoid Bioactivity The Journal of Clinical Endocrinology and Metabolism. ,vol. 88, pp. 323- 326 ,(2003) , 10.1210/JC.2002-020799

D Philibert, G Teutsch, RU 486 development Science. ,vol. 247, pp. 622- 622 ,(1990) , 10.1126/SCIENCE.2300819

LOUISA LAUE, MICHAEL T. LOTZE, GEORGE P. CHROUSOS, KEVIN BARNES, D. LYNN LORIAUX, THOMAS A. FLEISHER, Effect of Chronic Treatment with the Glucocorticoid Antagonist RU 486 in Man: Toxicity, Immunological, and Hormonal Aspects The Journal of Clinical Endocrinology and Metabolism. ,vol. 71, pp. 1474- 1480 ,(1990) , 10.1210/JCEM-71-6-1474

Ingrid Jung-Testas, Etienne-Emile Baulieu, Inhibition of glucocorticosteroid action in cultured L-929 mouse fibroblasts by RU 486, a new anti-glucocorticosteroid of high affinity for the glucocorticosteroid receptor. Experimental Cell Research. ,vol. 147, pp. 177- 182 ,(1983) , 10.1016/0014-4827(83)90282-3