Application of Plackett-Burman screening design for preparing glibenclamide nanoparticles for dissolution enhancement
作者： Sunny R Shah , Rajesh H Parikh , Jayant R Chavda , Navin R Sheth , None
DOI: 10.1016/J.POWTEC.2012.10.055
关键词: Solvent 、 Dissolution 、 Particle size 、 Chromatography 、 Regression analysis 、 Poloxamer 、 Surface-area-to-volume ratio 、 Plackett–Burman design 、 Chemistry 、 Pareto chart
摘要: This study is to improve the dissolution characteristics of a poorly water-soluble drug glibenclamide (GLB), by preparing nanoparticles through liquid anti solvent precipitation. A Plackett…
cheric.org
elsevier.com参考文章(21)
Min-Soo Kim, Shun-Ji Jin, Jeong-Soo Kim, Hee Jun Park, Ha-Seung Song, Reinhard H.H. Neubert, Sung-Joo Hwang, Preparation, characterization and in vivo evaluation of amorphous atorvastatin calcium nanoparticles using supercritical antisolvent (SAS) process. European Journal of Pharmaceutics and Biopharmaceutics. ,vol. 69, pp. 454- 465 ,(2008) , 10.1016/J.EJPB.2008.01.007
Yamasani Rao, Mittapalli Kumar, Shashank Apte, Formulation of Nanosuspensions of Albendazole for Oral Administration Current Nanoscience. ,vol. 4, pp. 53- 58 ,(2008) , 10.2174/157341308783591807
Dhananjay S. Singare, Seshasai Marella, K. Gowthamrajan, Giriraj T. Kulkarni, Rajesh Vooturi, Parchuri Srinivasa Rao, Optimization of formulation and process variable of nanosuspension: An industrial perspective International Journal of Pharmaceutics. ,vol. 402, pp. 213- 220 ,(2010) , 10.1016/J.IJPHARM.2010.09.041
Sudhir Verma, Bryan D. Huey, Diane J. Burgess, Scanning probe microscopy method for nanosuspension stabilizer selection. Langmuir. ,vol. 25, pp. 12481- 12487 ,(2009) , 10.1021/LA9016432
Neelam Seedher, Mamta Kanojia, Co-solvent solubilization of some poorly-soluble antidiabetic drugs Pharmaceutical Development and Technology. ,vol. 14, pp. 185- 192 ,(2009) , 10.1080/10837450802498894
Sudhir Verma, Rajeev Gokhale, Diane J. Burgess, A comparative study of top-down and bottom-up approaches for the preparation of micro/nanosuspensions. International Journal of Pharmaceutics. ,vol. 380, pp. 216- 222 ,(2009) , 10.1016/J.IJPHARM.2009.07.005
Ugo Bilati, Eric Allémann, Eric Doelker, Development of a nanoprecipitation method intended for the entrapment of hydrophilic drugs into nanoparticles. European Journal of Pharmaceutical Sciences. ,vol. 24, pp. 67- 75 ,(2005) , 10.1016/J.EJPS.2004.09.011
Sachin Kumar Singh, K.K. Srinivasan, K. Gowthamarajan, Dhananjay S. Singare, Dev Prakash, Narayan Babulal Gaikwad, Investigation of preparation parameters of nanosuspension by top-down media milling to improve the dissolution of poorly water-soluble glyburide. European Journal of Pharmaceutics and Biopharmaceutics. ,vol. 78, pp. 441- 446 ,(2011) , 10.1016/J.EJPB.2011.03.014
S. Otoom, M. Hasan, N. Najib, The bioavailability of glyburide (glibenclamide) under fasting and feeding conditions: a comparative study International Journal of Pharmaceutical Medicine. ,vol. 15, pp. 117- 120 ,(2001) , 10.1097/00124363-200106000-00003
Marc Lindenberg, Sabine Kopp, Jennifer B Dressman, Classification of orally administered drugs on the World Health Organization Model list of Essential Medicines according to the biopharmaceutics classification system. European Journal of Pharmaceutics and Biopharmaceutics. ,vol. 58, pp. 265- 278 ,(2004) , 10.1016/J.EJPB.2004.03.001