New strategies towards proline derivatives as conformationally constrained arginine analogues
作者： Nadia Pellegrini , Martine Schmitt , Sébastien Guery , Jean-Jacques Bourguignon
DOI: 10.1016/S0040-4039(02)00424-0
关键词: Chemistry 、 Proline 、 Pyrrolidine 、 Arginine 、 Organic chemistry 、 Stereochemistry
摘要: Abstract The cyano derivatives of 3-functionalized dehydroprolines led to arginine semi–constrained analogues.
elsevier.com
sci-hub.se 参考文章(15)
Marcos JoséS. Carpes, Paulo Cesar M.L. Miranda, Carlos Roque D. Correia, STEREOSELECTIVE SYNTHESIS OF CONFORMATIONALLY RESTRICTED ANALOGUES OF ASPARTIC AND GLUTAMIC ACIDS FROM ENDOCYCLIC ENECARBAMATES Tetrahedron Letters. ,vol. 38, pp. 1869- 1872 ,(1997) , 10.1016/S0040-4039(97)00238-4
Hiroshi Maeda, George A. Kraus, A Direct Route to Biologically Active Kainic Acid Analogs. Journal of Organic Chemistry. ,vol. 62, pp. 2314- 2315 ,(1997) , 10.1021/JO962114S
Qian Wang, N. AndréSasaki, Pierre Potier, ASYMMETRIC SYNTHESIS OF 4-SUBSTITUTED PROLINES AS CONFORMATIONALLY CONSTRAINED AMINO ACID ANALOGUES Tetrahedron. ,vol. 54, pp. 15759- 15780 ,(1998) , 10.1016/S0040-4020(98)00989-2
Dee W. Brooks, Keith W. Woods, Chiral building blocks for fused cyclopentanoids: enantioselective synthesis of 5-methylbicyclo[3.3.0]oct-1-ene-3,6-dione and derivatives Journal of Organic Chemistry. ,vol. 52, pp. 2036- 2039 ,(1987) , 10.1021/JO00386A026
John M. Matsoukas, Dimitris Panagiotopoulos, Maria Keramida, Thomas Mavromoustakos, Raghav Yamdagni, Qiao Wu, Graham J. Moore, Mahmoud Saifeddine, Morley D. Hollenberg, Synthesis and contractile activities of cyclic thrombin receptor-derived peptide analogues with a Phe-Leu-Leu-Arg motif: importance of the Phe/Arg relative conformation and the primary amino group for activity. Journal of Medicinal Chemistry. ,vol. 39, pp. 3585- 3591 ,(1996) , 10.1021/JM950690V
D. Damour, J.-P. Pulicani, M. Vuilhorgne, S. Mignani, cis- and trans-3-(3-Indolyl)proline Derivatives as Conformationally Restricted Analogues of Tryptophan Synlett. ,vol. 1999, pp. 786- 788 ,(1999) , 10.1055/S-1999-2708
Rui Zhang, Ahmed Mamai, Jose S. Madalengoitia, Cyclopropanation Reactions of Pyroglutamic Acid-Derived Synthons with Akylidene Transfer Reagents Journal of Organic Chemistry. ,vol. 64, pp. 547- 555 ,(1999) , 10.1021/JO9816109
Yasuji Yamada, Toshihide lshii, Masayuki Kimura, Kunio Hosaka, A direction controlled Dieckmann type cyclization of half-thiol diesters Tetrahedron Letters. ,vol. 22, pp. 1353- 1354 ,(1981) , 10.1016/S0040-4039(01)90316-8
Mukund P. Sibi, James W. Christensen, Sung-Gyu Kim, MariJean Eggen, Chad Stessman, Larry Oien, Chemoselective Dieckmann-like condensations using N-methoxy-N-methylamides Tetrahedron Letters. ,vol. 36, pp. 6209- 6212 ,(1995) , 10.1016/0040-4039(95)01251-C
Thomas R. Webb, Charles Eigenbrot, Conformationally restricted arginine analogs Journal of Organic Chemistry. ,vol. 56, pp. 3009- 3016 ,(1991) , 10.1021/JO00009A016