Iodine-catalyzed regioselective 2-sulfonylation of indoles with sodium sulfinates.
作者： Fuhong Xiao , Hui Chen , Hao Xie , Shuqing Chen , Luo Yang
DOI: 10.1021/OL402987U
关键词: Chemistry 、 Iodine 、 Metal catalyst 、 Regioselectivity 、 Catalysis 、 Organic chemistry 、 Indole formation 、 Sodium
摘要: Iodine-catalyzed selective 2-arylsulfonyl indole formation from indoles and sodium sulfinates is disclosed. Various substituted were obtained in one pot the absence of metal catalyst at room temperature under air.
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