Enantioselective synthesis of trifluoromethylated dihydroquinoxalinones via palladium-catalyzed hydrogenation
作者： Mu-Wang Chen , Zhihong Deng , Qin Yang , Jian Huang , Yiyuan Peng
DOI: 10.1039/C8QO01361F
关键词: Catalysis 、 Palladium 、 Asymmetric hydrogenation 、 Enantioselective synthesis 、 Combinatorial chemistry 、 Chemistry 、 Enantiomeric excess 、 Trifluoromethyl
摘要: … 3-(trifluoromethyl)-3,4-dihydroquinoxalinones with up to 99% ee. In addition, the 3-(trifluoromethyl)-3,4-dihydroquinoxalinones can be conveniently converted into 2-(trifluoromethyl)-1,2,…
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