Straightforward Approach Toward Dihydrothiazoles via Intramolecular Bromocyclization

作者: Seyed Esmail Sadat-Ebrahimi , Marzieh Ganjizadeh Zarj , Setareh Moghimi , Azadeh Yahya-Meymandi , Mohammad Mahdavi

DOI: 10.1080/00397911.2015.1067707

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摘要: AbstractAn intramolecular bromonium ion–assisted cyclization with sulfur as an internal nucleophile is described. Starting from benzoyl chlorides, this method provides easy procedure for the synthesis of dihydrothiazole derivatives in moderate to good yields.

参考文章(17)
Majid M. Heravi, Setareh Moghimi, An efficient synthesis of thiazol-2-imine derivatives via a one-pot, three-component reaction Tetrahedron Letters. ,vol. 53, pp. 392- 394 ,(2012) , 10.1016/J.TETLET.2011.11.017
Gordon W. Gribble, Naturally Occurring Organohalogen Compounds Accounts of Chemical Research. ,vol. 31, pp. 141- 152 ,(1998) , 10.1021/AR9701777
R.J. Baumann, G.D. Mayer, L.D. Fite, L.M. Gill, B.L. Harrison, In vitro and in vivo Candicidal Activities of 2-(p-n-Hexylphenylamino)-1,3-Thiazoline Chemotherapy. ,vol. 37, pp. 157- 165 ,(1991) , 10.1159/000238849
April L. Bernacki, Lingyang Zhu, D. David Hennings, A selective and convenient method for the synthesis of 2-phenylaminothiazolines. Organic Letters. ,vol. 12, pp. 5526- 5529 ,(2010) , 10.1021/OL102428M
John W. Reynolds, XV.—On “propylene,” a new hydrocarbon of the series CnHn Q. J. Chem. Soc.. ,vol. 3, pp. 111- 120 ,(1851) , 10.1039/QJ8510300111
Souad Kasmi, Jack Hamelin, Hadj Benhaoua, Microwave-assisted solvent-free synthesis of iminothiazolines Tetrahedron Letters. ,vol. 39, pp. 8093- 8096 ,(1998) , 10.1016/S0040-4039(98)01836-X
Jing Wang, Hai-Bo Liu, Wei Wang, Il Kim, Chang-Sik Ha, A thiazoline-containing cobalt(II) complex based colorimetric fluorescent probe: “turn-on” detection of fluoride Dalton Transactions. pp. 10422- 10425 ,(2009) , 10.1039/B918887H
Behnaz Shafii, Mina Saeedi, Mohammad Mahdavi, Alireza Foroumadi, Abbas Shafiee, Novel Four-Step Synthesis of Thioxo-quinazolino[3,4-a]quinazolinone Derivatives Synthetic Communications. ,vol. 44, pp. 215- 221 ,(2014) , 10.1080/00397911.2013.800211
D. Christopher Braddock, Stephen A. Hermitage, Lilian Kwok, Rebecca Pouwer, Joanna M. Redmond, Andrew J. P. White, The generation and trapping of enantiopure bromonium ions Chemical Communications. pp. 1082- 1084 ,(2009) , 10.1039/B816914D