AAZTA5-squaramide ester competing with DOTA-, DTPA- and CHX-A″-DTPA-analogues: Promising tool for 177Lu-labeling of monoclonal antibodies under mild conditions.

作者: Frank Rösch , Benedikt Klasen , Euy Sung Moon

DOI: 10.1016/J.NUCMEDBIO.2021.03.007

关键词:

摘要: … Coupling of AAZTA 5 -SA to the monoclonal antibody bevacizumab allowed for 177 Lu-… 177 Lu-labeling of sensitive biomolecules such as antibodies for theranostic applications. …

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