Structural requirements of KTS-disintegrins for inhibition of α1β1 integrin
作者： Meghan C. Brown , Johannes A. Eble , Juan J. Calvete , Cezary Marcinkiewicz
DOI: 10.1042/BJ20081403
关键词:
摘要: … The potency of recombinant KTS-disintegrins also depended on the residue C-terminally adjacent to the active motif. Substitution of Leu 24 of wild-type obtustatin for an alanine residue …
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