Direct salinization of trelagliptin from solid forms by mechanochemistry and its mechanism of salt formation
作者： Kailin Xu , Menglin Qian , Jiewu Leng , Jie Bai , Qinglan Li
DOI: 10.1039/D0CE00984A
关键词:
摘要: … In this study, an efficient mechanochemical salinization method was developed to prepare trelagliptin succinate (TRE-S), the first once-weekly oral treatment drug for type II diabetes. …
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