2[prime] and 3[prime] Carboranyl uridines and their diethyl ether adducts

摘要: A process is described for preparing carboranyl uridine nucleoside compounds and their diethyl ether adducts, which exhibit a tenfold increase in boron content over prior art containing compounds. The enhanced lipophilicity hydrophilic properties adequate to enable solvation aqueous media subsequent incorporation of the methods neutron capture therapy mammalian tumor cells. No Drawings