Medicinal chemistry strategies to discover P-glycoprotein inhibitors: An update.
作者： Jinyun Dong , Zuodong Qin , Wei-Dong Zhang , Gang Cheng , Assaraf G. Yehuda
DOI: 10.1016/J.DRUP.2020.100681
关键词:
摘要: … Herein, we provide a comprehensive review of the synthetic and natural products that have … The present review focuses primarily on the structural features, design strategies, and …
sci-hub.se 参考文章(229)
Stéphane ORLOWSKI, Lluis M. MIR, Jean BELEHRADEK, Manuel GARRIGOS, Effects of steroids and verapamil on P-glycoprotein ATPase activity: progesterone, desoxycorticosterone, corticosterone and verapamil are mutually non-exclusive modulators Biochemical Journal. ,vol. 317, pp. 515- 522 ,(1996) , 10.1042/BJ3170515
C P H Yang, S G DePinho, L M Greenberger, R J Arceci, S B Horwitz, Progesterone interacts with P-glycoprotein in multidrug-resistant cells and in the endometrium of gravid uterus. Journal of Biological Chemistry. ,vol. 264, pp. 782- 788 ,(1989) , 10.1016/S0021-9258(19)85010-X
Raymond P. Perez, Thomas C. Hamilton, Robert F. Ozols, Robert C. Young, Mechanisms and modulation of resistance to chemotherapy in ovarian cancer. Cancer. ,vol. 71, pp. 1571- 1580 ,(1993) , 10.1002/CNCR.2820710424
G D Eytan, M J Borgnia, R Regev, Y G Assaraf, Transport of polypeptide ionophores into proteoliposomes reconstituted with rat liver P-glycoprotein. Journal of Biological Chemistry. ,vol. 269, pp. 26058- 26065 ,(1994) , 10.1016/S0021-9258(18)47159-1
Di Chen, Sheng Biao Wan, Huanjie Yang, Jian Yuan, Tak Hang Chan, Q. Ping Dou, EGCG, GREEN TEA POLYPHENOLS AND THEIR SYNTHETIC ANALOGS AND PRODRUGS FOR HUMAN CANCER PREVENTION AND TREATMENT Advances in Clinical Chemistry. ,vol. 53, pp. 155- 177 ,(2011) , 10.1016/B978-0-12-385855-9.00007-2
Tripta Bansal, Manu Jaggi, Roop Khar, Sushama Talegaonkar, Emerging significance of flavonoids as P-glycoprotein inhibitors in cancer chemotherapy. Journal of Pharmacy and Pharmaceutical Sciences. ,vol. 12, pp. 46- 78 ,(2009) , 10.18433/J3RC77
Chiara Riganti, Costanzo Costamagna, Amalia Bosia, Dario Ghigo, Gianpiero Pescarmona, Erica Miraglia, Daniele Viarisio, Nitric oxide reverts the resistance to doxorubicin in human colon cancer cells by inhibiting the drug efflux. Cancer Research. ,vol. 65, pp. 516- 525 ,(2005)
Tae‐Eun Kim, Howard Lee, Kyoung Soo Lim, SeungHwan Lee, Seo‐Hyun Yoon, Kyung‐Mi Park, Hyesun Han, Sang‐Goo Shin, In‐Jin Jang, Kyung‐Sang Yu, Joo‐Youn Cho, None, Effects of HM30181, a P‐glycoprotein inhibitor, on the pharmacokinetics and pharmacodynamics of loperamide in healthy volunteers British Journal of Clinical Pharmacology. ,vol. 78, pp. 556- 564 ,(2014) , 10.1111/BCP.12368
Grégory Gatouillat, Abdulmagid Alabdul Magid, Eric Bertin, Hassan El btaouri, Hamid Morjani, Catherine Lavaud, Claudie Madoulet, Medicarpin and millepurpan, two flavonoids isolated from Medicago sativa, induce apoptosis and overcome multidrug resistance in leukemia P388 cells Phytomedicine. ,vol. 22, pp. 1186- 1194 ,(2015) , 10.1016/J.PHYMED.2015.09.005
R. S. Lewis, J. Fidel, S. Dassanayake, M. H. Court, N. S. Burke, K. L. Mealey, Comparison of chemotherapeutic drug resistance in cells transfected with canine ABCG2 or feline ABCG2 Veterinary and Comparative Oncology. ,vol. 15, pp. 411- 420 ,(2017) , 10.1111/VCO.12177