A newly synthesized selective casein kinase I inhibitor, N-(2-aminoethyl)-5-chloroisoquinoline-8-sulfonamide, and affinity purification of casein kinase I from bovine testis.
作者： T Chijiwa , M Hagiwara , H Hidaka
DOI: 10.1016/S0021-9258(18)83679-1
关键词:
摘要: When screening various isoquinolinesulfonamide compounds which we synthesized, CKI-7, N-(2-amino-ethyl)-5-chloroisoquinoline-8-sulfonamide, was found to have a potent …
sci-hub.st 参考文章(22)
M.E. Dahmus, Purification and properties of calf thymus casein kinases I and II. Journal of Biological Chemistry. ,vol. 256, pp. 3319- 3325 ,(1981) , 10.1016/S0021-9258(19)69609-2
GARY M. HATHAWAY, JOLINDA A. TRAUGH, Casein kinases--multipotential protein kinases. Current Topics in Cellular Regulation. ,vol. 21, pp. 101- 127 ,(1982) , 10.1016/B978-0-12-152821-8.50009-8
Hiroyoshi Hidaka, Toshio Tanaka, [44] Transmembrane Ca2+ signaling and a new class of inhibitors Methods in Enzymology. ,vol. 139, pp. 570- 582 ,(1987) , 10.1016/0076-6879(87)39113-X
K.M. Rose, L.E. Bell, D.A. Siefken, S.T. Jacob, A heparin-sensitive nuclear protein kinase. Purification, properties, and increased activity in rat hepatoma relative to liver. Journal of Biological Chemistry. ,vol. 256, pp. 7468- 7477 ,(1981) , 10.1016/S0021-9258(19)68986-6
T L McGuinness, Y Lai, P Greengard, Ca2+/calmodulin-dependent protein kinase II. Isozymic forms from rat forebrain and cerebellum. Journal of Biological Chemistry. ,vol. 260, pp. 1696- 1704 ,(1985) , 10.1016/S0021-9258(18)89650-8
E Itarte, K P Huang, Purification and properties of cyclic AMP-independent glycogen synthase kinase 1 from rabbit skeletal muscle. Journal of Biological Chemistry. ,vol. 254, pp. 4052- 4057 ,(1979) , 10.1016/S0021-9258(18)50694-3
G.M. Hathaway, J.A. Traugh, Cyclic nucleotide-independent protein kinases from rabbit reticulocytes. Purification of casein kinases. Journal of Biological Chemistry. ,vol. 254, pp. 762- 768 ,(1979) , 10.1016/S0021-9258(17)37871-7
G.M. Hathaway, T.H. Lubben, J.A. Traugh, Inhibition of casein kinase II by heparin. Journal of Biological Chemistry. ,vol. 255, pp. 8038- 8041 ,(1980) , 10.1016/S0021-9258(19)70601-2
K P Huang, E Itarte, T J Singh, A Akatsuka, Phosphorylation of glycogen synthase by cyclic AMP-independent casein kinase-2 from rabbit skeletal muscle. Journal of Biological Chemistry. ,vol. 257, pp. 3236- 3242 ,(1982) , 10.1016/S0021-9258(19)81101-8
F Meggio, F Marchiori, G Borin, G Chessa, L A Pinna, Synthetic peptides including acidic clusters as substrates and inhibitors of rat liver casein kinase TS (type-2). Journal of Biological Chemistry. ,vol. 259, pp. 14576- 14579 ,(1984) , 10.1016/S0021-9258(17)42640-8