The Synthesis of 5-Substituted-2, 4-dimethoxypyrimidines and Some Related Nucleoside Analogues
作者： R. F. Whale , P. L. Coe , R. T. Walker
DOI: 10.1080/07328319208021184
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摘要: Abstract The reaction of 5-formyl-2,4-dimethoxypyrimidine with active methylene compounds in the Knoevenagel and subsequent nucleoside formation reactions some products was investigated. A new synthesis (E)-5-(2-bromovinyl)uracil an improved 5-formyl-2′,3′-isopropylidene uridine are reported.
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