Benzamide derivatives and their use as vasopressin antagonists
作者： Hiroyuki Setoi , Tatsuya Zenkoh , Kentaro Sato , Hirokazu Tanaka , Hitoshi Sawada
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摘要: This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc., and represented by general formula (I), wherein R1 is aryl optionally substituted with lower alkoxy, R2 alkyl, R3 hydrogen, R4 R5 A NH, E (a), X -CH=CH-, -CH=N-, or S, Y CH N, pharmaceutically acceptable salts thereof, processes for preparation thereof pharmaceutical composition comprising the same.
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