Azaindoles. LXIV. Search for β-adrenoblockers in the 5-azaindole series

Robert C. Tarazi, Harriet P. Dustan, Beta adrenergic blockade in hypertension The American Journal of Cardiology. ,vol. 29, pp. 633- 640 ,(1972) , 10.1016/0002-9149(72)90164-6

Leonard M. Weinstock, Dennis M. Mulvey, Roger. Tull, Synthesis of the .beta.-adrenergic blocking agent timolol from optically active precursors Journal of Organic Chemistry. ,vol. 41, pp. 3121- 3124 ,(1976) , 10.1021/JO00881A011

Hendrika J. Waal-Manning, Hypertension: which beta-blocker? Drugs. ,vol. 12, pp. 412- 441 ,(1976) , 10.2165/00003495-197612060-00002

Johannes Smid, Die Struktur solvatisierter Ionenpaare Angewandte Chemie. ,vol. 84, pp. 127- 144 ,(1972) , 10.1002/ANGE.19720840402

John J. Baldwin, Edward L. Engelhardt, Ralph Hirschmann, Gerald S. Ponticello, Joseph G. Atkinson, Burton K. Wasson, Charles S. Sweet, Alexander Scriabine, Heterocyclic analogues of the antihypertensive beta-adrenergic blocking agent (S)-2-[3-(ter-butylamino)-2-hydroxypropoxy]-3-cyanopyridine. Journal of Medicinal Chemistry. ,vol. 23, pp. 65- 70 ,(1980) , 10.1021/JM00175A012

William E. Kreighbaum, W. Lesley Matier, Ronald D. Dennis, Joseph L. Minielli, David Deitchman, James L. Perhach, William T. Comer, Antihypertensive indole derivatives of phenoxypropanolamines with beta-adrenergic receptor antagonist and vasodilating activity. Journal of Medicinal Chemistry. ,vol. 23, pp. 285- 289 ,(1980) , 10.1021/JM00177A015

G.L. Wollam, R.W. Gifford, R.C. Tarazi, Antihypertensive drugs: clinical pharmacology and therapeutic use. Drugs. ,vol. 14, pp. 420- 460 ,(1977) , 10.2165/00003495-197714060-00002