Metalation of Pyridazine, Cinnoline, and Phthalazine
作者： Ernst Horkel
DOI: 10.1007/7081_2012_97
关键词:
摘要: This chapter reviews the metalation of pyridazine, cinnoline, and phthalazine derivatives as well usage hereby formed organometallic compounds in subsequent reactions. The main topics under discussion are lithiation, magnesation, zincation, focus being on deprotonative by properly chosen strong bases, e.g. lithiumdiisopropylamide or lithium 2,2,6,6-tetramethylpiperidide. A short upon boronyl stannyl three diazines investigation is enclosed at end chapter.
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