Serine protease inhibitors

作者: Bohdan Waszkowycz , Christopher Neil Farthing , Sarah Elizabeth Lively , Martin James Harrison , Keith Michael Johnson

DOI:

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摘要: Compounds having structure (A) are useful to inhibit serine protease enzymes, such as TF/factor VIIa, factor Xa, thrombin and kallikrein. These compounds may be used in methods of preventing and/or treating clotting disorders.

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