Synthesis of Thioamides by Catalyst‐Free Three‐Component Reactions in Water

作者: Hualong Xu , Hang Deng , Zhengkai Li , Haifeng Xiang , Xiangge Zhou

DOI: 10.1002/EJOC.201301148

关键词:

摘要: Three-component reactions involving amines, aldehydes, and elemental sulfur powder are reported to afford thioamides in a simple one-pot procedure the absence of catalyst. A variety can be obtained good excellent yields up 88 %.

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