The first carboranyl bis(adenosine diphosphate) (CBADP): a synthetic investigation
作者： Kamesh Vyakaranam , Geeta Rana , Shannon Delaney , Sarah Ledger , Narayan S. Hosmane
DOI: 10.1016/S1387-7003(03)00067-4
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摘要: Abstract The synthesis of the first carboranyl bis(adenosine diphosphate) (CBADP) ( 5 ) was achieved in three steps. step involved reaction o -carborane dianion, 1 , with methyl dichlorophosphate to yield 2 . Reagent 4 synthesized by bis-benzoyl-protected adenosine phosphoryl chloride, followed protection free hydroxyl group product, 3 triflate. final converged both and into title compound, CBADP ).
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