Boron-based small molecules in disease detection and treatment (2013–2016)

Takumi Watanabe, Hikaru Abe, Isao Momose, Yoshikazu Takahashi, Daishiro Ikeda, Yuzuru Akamatsu, Structure-activity relationship of boronic acid derivatives of tyropeptin: proteasome inhibitors. Bioorganic & Medicinal Chemistry Letters. ,vol. 20, pp. 5839- 5842 ,(2010) , 10.1016/J.BMCL.2010.07.122

Scott J. Hecker, K. Raja Reddy, Maxim Totrov, Gavin C. Hirst, Olga Lomovskaya, David C. Griffith, Paula King, Ruslan Tsivkovski, Dongxu Sun, Mojgan Sabet, Ziad Tarazi, Matthew C. Clifton, Kateri Atkins, Amy Raymond, Kristy T. Potts, Jan Abendroth, Serge H. Boyer, Jeffrey S. Loutit, Elizabeth E. Morgan, Stephanie Durso, Michael N. Dudley, Discovery of a Cyclic Boronic Acid β-Lactamase Inhibitor (RPX7009) with Utility vs Class A Serine Carbapenemases. Journal of Medicinal Chemistry. ,vol. 58, pp. 3682- 3692 ,(2015) , 10.1021/ACS.JMEDCHEM.5B00127

Zerrin Canturk, Yağmur Tunali, Seval Korkmaz, Zafer Gulbaş, Cytotoxic and apoptotic effects of boron compounds on leukemia cell line Cytotechnology. ,vol. 68, pp. 87- 93 ,(2016) , 10.1007/S10616-014-9755-7

D Raddatz, G Ramadori, Carbohydrate metabolism and the liver: actual aspects from physiology and disease. Zeitschrift Fur Gastroenterologie. ,vol. 45, pp. 51- 62 ,(2007) , 10.1055/S-2006-927394

Priscila Milani, Marilene Demasi, Leandro de Rezende, Antonia T.-do Amaral, Leandro H. Andrade, Synthesis ofl-cysteine-based boron compounds and their evaluation as proteasome inhibitors New J. Chem.. ,vol. 38, pp. 4859- 4871 ,(2014) , 10.1039/C4NJ00612G

Julie I. Jay, Bonnie E. Lai, David G. Myszka, Alamelu Mahalingam, Kris Langheinrich, David F. Katz, Patrick F. Kiser, Multivalent benzoboroxole functionalized polymers as gp120 glycan targeted microbicide entry inhibitors Molecular Pharmaceutics. ,vol. 7, pp. 116- 129 ,(2010) , 10.1021/MP900159N

Julie Arnaud, Aymeric Audfray, Anne Imberty, Binding sugars: from natural lectins to synthetic receptors and engineered neolectins Chemical Society Reviews. ,vol. 42, pp. 4798- 4813 ,(2013) , 10.1039/C2CS35435G

H. Fu, H. Fang, Jie Sun, H. Wang, A. Liu, J. Sun, Z. Wu, Boronic Acid-based Enzyme Inhibitors: A Review of Recent Progress Current Medicinal Chemistry. ,vol. 21, pp. 3271- 3280 ,(2014) , 10.2174/0929867321666140601200803

Jun Yan, Greg Springsteen, Susan Deeter, Binghe Wang, The relationship among pKa, pH, and binding constants in the interactions between boronic acids and diols—it is not as simple as it appears Tetrahedron. ,vol. 60, pp. 11205- 11209 ,(2004) , 10.1016/J.TET.2004.08.051

Tsutomu Akama, Chen Dong, Charlotte Virtucio, Yvonne R. Freund, Daitao Chen, Matthew D. Orr, Robert T. Jacobs, Yong-Kang Zhang, Vincent Hernandez, Yang Liu, Anne Wu, Wei Bu, Liang Liu, Kurt Jarnagin, Jacob J. Plattner, Discovery and structure-activity relationships of 6-(benzoylamino)benzoxaboroles as orally active anti-inflammatory agents. Bioorganic & Medicinal Chemistry Letters. ,vol. 23, pp. 5870- 5873 ,(2013) , 10.1016/J.BMCL.2013.08.096