Inhibition of Cell Division and Stimulation of Progesterone Receptor Synthesis in Rat Oestrogen Target Tissues by Non-Steroidal Antioestrogens
作者： V. C. Jordan , C. J. Dix , G. Prestwich
DOI: 10.1007/978-1-4757-6589-2_7
关键词:
摘要: Tamoxifen and monohydroxytamoxifen (Fig. 1) are non-steroidal compounds that antagonise the effects of oestradiol in rat (1–4). However, although they antioestrogenic also possess atypical oestrogenic activity probably best described as partial agonists.
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