seco-C/D ring analogues of ergot alkaloids. Synthesis via intramolecular Heck and ring-closing metathesis reactions.

作者: Alexey V. Kalinin , Brian A. Chauder , Suman Rakhit , Victor Snieckus

DOI: 10.1021/OL035398T

关键词:

摘要: Intramolecular Heck and ring-closing metathesis reactions on key intermediates 10 15, respectively, provide efficient entries into seco-C/D ring analogues of Ergot alkaloids 12 16, compounds potential synthetic biological interest.

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