Discovery of highly potent triazole antifungal derivatives by heterocycle-benzene bioisosteric replacement.
作者： Zhigan Jiang , Yan Wang , Wenya Wang , Shengzheng Wang , Bo Xu
DOI: 10.1016/J.EJMECH.2013.04.025
关键词:
摘要: On the basis of our previously discovered triazole antifungal lead compounds, heterocycle-benzene bioisosteric replacement was used to improve their pharmacokinetic profile. The …
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