Chemistry of folic acid antagonists (a review)

作者: M. P. Nemeryuk , M. V. Pykhova , T. S. Safonova

DOI: 10.1007/BF00763372

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参考文章(97)
Joseph I. DeGraw, Roy L. Kisliuk, Yvette Gaumont, Charles M. Baugh, Antimicrobial activity of 8-deazafolic acid. Journal of Medicinal Chemistry. ,vol. 17, pp. 470- 471 ,(1974) , 10.1021/JM00250A026
J. R. Piper, G. S. McCaleb, J. A. Montgomery, Roy L. Kisliuk, Y. Gaumont, F. M. Sirotnak, 10-Propargylaminopterin and alkyl homologs of methotrexate as inhibitors of folate metabolism Journal of Medicinal Chemistry. ,vol. 25, pp. 877- 880 ,(1982) , 10.1021/JM00349A024
William W. Lee, Abelardo P. Martinez, Leon Goodman, Folic acid antagonists. Methotrexate analogs containing spurious amino acids. Dichlorohomofolic acid. Journal of Medicinal Chemistry. ,vol. 17, pp. 326- 330 ,(1974) , 10.1021/JM00249A015
M. G. Nair, Shiang-Yuan Chen, Roy L. Kisliuk, Y. Gaumont, D. Strumpf, Folate analogues altered in the C9-N10 bridge region: 11-thiohomofolic acid. Journal of Medicinal Chemistry. ,vol. 22, pp. 850- 855 ,(1979) , 10.1021/JM00193A019
James C. Parham, Mary Agnes Templeton, Paul L. Chello, Francis M. Sirotnak, Synthesis and Properties of 10-Benzylaminopterin Journal of Heterocyclic Chemistry. ,vol. 16, pp. 1645- 1646 ,(1979) , 10.1002/JHET.5570160826
Terence R. Jones, 5-Substituted quinazoline antifolates European Journal of Cancer (1965). ,vol. 16, pp. 707- 711 ,(1980) , 10.1016/0014-2964(80)90213-3
Yu-Uji Nakahara, Isao Sekikawa, Shichiro Kakimoto, Synthesis of N-([2-([(2-amino-3,4-dihydro-4-oxo-6-pteridinyl)methyl]amino)-5- pyrazinyl]carbonyl)-L-glutamic acid (2′,5′-diazafolic acid) Journal of Heterocyclic Chemistry. ,vol. 12, pp. 1073- 1074 ,(1975) , 10.1002/JHET.5570120558
Andre Rosowsky, Ronald Forsch, Jack Uren, Michael Wick, Methotrexate analogs. 14. Synthesis of new .gamma.-substituted derivatives as dihydrofolate reductase inhibitors and potential anticancer agents Journal of Medicinal Chemistry. ,vol. 24, pp. 1450- 1455 ,(1981) , 10.1021/JM00144A016
Dan Carol Suster, Eutanta Tarnauceanu, Dumitru Ionescu, Vasile Dobre, Ion Niculescu-Duvaz, Potential anticancer agents. 16. Methotrexate analogs with a modified peptide side chain Journal of Medicinal Chemistry. ,vol. 21, pp. 1162- 1165 ,(1978) , 10.1021/JM00209A015
Edward C. Taylor, Peter J. Harrington, Stephen R. Fletcher, G. Peter Beardsley, Richard G. Moran, Synthesis of the antileukemic agents 5,10-dideazaaminopterin and 5,10-dideaza-5,6,7,8-tetrahydroaminopterin. Journal of Medicinal Chemistry. ,vol. 28, pp. 914- 921 ,(1985) , 10.1021/JM00145A012