Discovery of Antimalarial Drug Artemisinin and Beyond

作者: Weiwei Mao , Yu Zhang , Ao Zhang

DOI: 10.1002/9781118219683.CH10

关键词:

摘要: … useful for treating a variety of diseases were isolated including anticancer agents (taxol, doxorubicin, and camptothecin), lipid control drugs of which lovastatin, atorvastatin, fluvastatin, …

参考文章(130)
Louis Koné Penali, Frans Herwig Jansen, Single-day, three-dose treatment with fixed dose combination artesunate/sulfamethoxypyrazine/pyrimethamine to cure Plasmodium falciparum malaria International Journal of Infectious Diseases. ,vol. 12, pp. 430- 437 ,(2008) , 10.1016/J.IJID.2007.12.006
Stephen Hindley, Stephen A Ward, Richard C Storr, Natalie L Searle, Patrick G Bray, B Kevin Park, Jill Davies, Paul M O'Neill, None, Mechanism-based design of parasite-targeted artemisinin derivatives: synthesis and antimalarial activity of new diamine containing analogues. Journal of Medicinal Chemistry. ,vol. 45, pp. 1052- 1063 ,(2002) , 10.1021/JM0109816
Ignacio Fita, Michael G. Rossmann, The active center of catalase Journal of Molecular Biology. ,vol. 185, pp. 21- 37 ,(1985) , 10.1016/0022-2836(85)90180-9
Mankil Jung, Xun Li, Daniel A Bustos, Hala N ElSohly, James D McChesney, A short and stereospecific synthesis of (+)-deoxoartemisinin and (−)-deoxodesoxyartemisinin Tetrahedron Letters. ,vol. 30, pp. 5973- 5976 ,(1989) , 10.1016/S0040-4039(01)93831-6
D. Klayman, Qinghaosu (artemisinin): an antimalarial drug from China Science. ,vol. 228, pp. 1049- 1055 ,(1985) , 10.1126/SCIENCE.3887571
Mai M Al-Oqail, Ahmed M Galal, Mohamed S Ahmad, Ahlam M Al-Fishawi, Farouk S El-Feraly, None, New Bioactive Azaartemisinin Derivatives Molecules. ,vol. 8, pp. 901- 909 ,(2003) , 10.3390/81200901
Richard K. Haynes, Wing-Yan Ho, Ho-Wai Chan, Burkhard Fugmann, Jörg Stetter, Simon L. Croft, Livia Vivas, Wallace Peters, Brian L. Robinson, Highly Antimalaria-Active Artemisinin Derivatives: Biological Activity Does Not Correlate with Chemical Reactivity Angewandte Chemie International Edition. ,vol. 43, pp. 1381- 1385 ,(2004) , 10.1002/ANIE.200352343
T K Dien, P J de Vries, N X Khanh, R Koopmans, L N Binh, D D Duc, P A Kager, C J van Boxtel, Effect of food intake on pharmacokinetics of oral artemisinin in healthy Vietnamese subjects. Antimicrobial Agents and Chemotherapy. ,vol. 41, pp. 1069- 1072 ,(1997) , 10.1128/AAC.41.5.1069
Richard K. Haynes, Ho-Wai Chan, Man-Ki Cheung, Shuk Ting Chung, Wai-Lun Lam, Hing-Wo Tsang, Arnd Voerste, Ian D. Williams, Stereoselective Preparation of 10α- and 10β-Aryl Derivatives of Dihydroartemisinin European Journal of Organic Chemistry. ,vol. 2003, pp. 2098- 2114 ,(2003) , 10.1002/EJOC.200300064
M V Vugt, B Gemperli, N J White, A Brockman, S Looareesuwan, I Gathmann, F Nosten, C Luxemburger, L Phaipun, P Wilairatana, Efficacy of six doses of artemether-lumefantrine (benflumetol) in multidrug-resistant Plasmodium falciparum malaria. American Journal of Tropical Medicine and Hygiene. ,vol. 60, pp. 936- 942 ,(1999) , 10.4269/AJTMH.1999.60.936