Processes and intermediates for preparing cysteine protease inhibitors

Tatsuya Shono, Naoki Kise, Akira Yamazaki, Hiroshi Ohmizu, Novel selective synthesis of α-chloromethyl, α,α-dichloromethyl, and α,α,α-trichloromethyl ketones from aldehyde utilizing electroreduction as key reactions Tetrahedron Letters. ,vol. 23, pp. 1609- 1612 ,(1982) , 10.1016/S0040-4039(00)87171-3

Xavier Creary, Elizabeth A. Burtch, Remarkably facile solvolyses of triflates via carbocationic processes in dimethyl sulfoxide. Journal of Organic Chemistry. ,vol. 69, pp. 1227- 1234 ,(2004) , 10.1021/JO0356558

Denice Mary Spero, Younes Bekkali, Yancey D. Ward, David S. Thomson, Sanxing Sun, Erick R. R. Young, Weimin Liu, Usha R. Patel, Eugene R. Hickey, Compounds useful as reversible inhibitors of cysteine proteases ,(2002)

Michel Therien, Christopher I. Bayly, Vouy Linh Truong, Jacques Yves Gauthier, Serge Leger, Cameron Black, Chun Sing Li, Christophe Mellon, Cheuk K. Lau, James T. Palmer, Michael J. Green, James W. Janc, Bernard Hirschbein, Dan Mckay, Chitra Baskaran, Cathepsin cysteine protease inhibitors ,(2003)

R Anilkumar, Donald J Burton, A highly efficient room temperature non-organometallic route for the synthesis of α,β,β-trifluorostyrenes by dehydrohalogenation Tetrahedron Letters. ,vol. 44, pp. 6661- 6664 ,(2003) , 10.1016/S0040-4039(03)01628-9

Brindaban C. Ranu, Sampak Samanta, Arijit Das, Reduction of trihalomethyl carbinols and their acetates, mesylates and tosylates by indium metal Tetrahedron Letters. ,vol. 43, pp. 5993- 5995 ,(2002) , 10.1016/S0040-4039(02)01262-5

Michael Stewart Large, Craig Johnstone, Howard Tucker, Philip Neil Edwards, John Oldfield, Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s ,(2000)