Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line.

作者: Carsten Uhd Nielsen , Claudiu T. Supuran , Andrea Scozzafava , Sven Frokjaer , Bente Steffansen

DOI: 10.1023/A:1020306926419

关键词:

摘要: Purpose. The aim of the present study was to evaluate whether transepithelial transport anticancer compound 4-toluenesulfonylureido-carnosine (Ts-carnosine) and dipeptide moiety L-carnosine due a hPepT1 carrier-mediated flux.

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