Metal-free direct regioselective thiolation of imidazoheterocycles in water at room temperature
作者： Dulin Kong , Qinghe Wang , Tiao Huang , Min Liang , Qiang Lin
DOI: 10.1016/J.TET.2019.01.059
关键词:
摘要: Abstract A metal-free direct thiolation of imidazoheterocycles with various thiophenol in water at room temperature has been developed. In addition, the chemistry provides several advantages including mild condition, high yields, good functional group tolerance, green solvents and suitable for large-scale operations.
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