An Overview of Recent Advances in Biological and Pharmaceutical Developments of Fluoro-containing Drugs

Hans‐Joachim Böhm, David Banner, Stefanie Bendels, Manfred Kansy, Bernd Kuhn, Klaus Müller, Ulrike Obst‐Sander, Martin Stahl, Fluorine in medicinal chemistry. Progress in Medicinal Chemistry. ,vol. 54, pp. 65- 133 ,(2015) , 10.1016/BS.PMCH.2014.11.001

Sanjeeva J. Wijeyesakere, Faik A. Nasser, Jeff W. Kampf, Alexey Y. Aksinenko, Vladimir B. Sokolov, Vladimir V. Malygin, Galina F. Makhaeva, Rudy J. Richardson, Diethyl [2,2,2-trifluoro-1-phenyl-sulfonyl-amino-1-(trifluoro-meth-yl)eth-yl]phospho-nate. Acta Crystallographica Section E-structure Reports Online. ,vol. 64, ,(2008) , 10.1107/S1600536808020175

Shengnan Ma, Jie Zhou, Aisha Roshan Mohamed Wali, Yiyan He, Xianghui Xu, James Zhenggui Tang, Zhongwei Gu, Self-assembly of pH-sensitive fluorinated peptide dendron functionalized dextran nanoparticles for on-demand intracellular drug delivery Journal of Materials Science: Materials in Medicine. ,vol. 26, pp. 219- ,(2015) , 10.1007/S10856-015-5550-Z

R. E. Banks, Fluorine chemistry at the millennium : fascinated by fluorine Elsevier. ,(2000)

Iwao Ojima, Fluorine in medicinal chemistry and chemical biology Wiley. ,(2009) , 10.1002/9781444312096

Miriam Benezra, Dolores Hambardzumyan, Oula Penate-Medina, Darren R. Veach, Nagavarakishore Pillarsetty, Peter Smith-Jones, Evan Phillips, Tatsuya Ozawa, Pat B. Zanzonico, Valerie Longo, Eric C. Holland, Steven M. Larson, Michelle S. Bradbury, Fluorine-labeled Dasatinib Nanoformulations as Targeted Molecular Imaging Probes in a PDGFB-driven Murine Glioblastoma Model Neoplasia. ,vol. 14, pp. 1132- 1143 ,(2012) , 10.1593/NEO.121750

Maria V. Papadopoulou, William D. Bloomer, Howard S. Rosenzweig, Ivan P. O’Shea, Shane R. Wilkinson, Marcel Kaiser, Eric Chatelain, Jean-Robert Ioset, Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation Bioorganic & Medicinal Chemistry. ,vol. 23, pp. 6467- 6476 ,(2015) , 10.1016/J.BMC.2015.08.014

Li-Yuan Zhang, Bao-Lei Wang, Yi-Zhou Zhan, Yan Zhang, Xiao Zhang, Zheng-Ming Li, Synthesis and biological activities of some fluorine- and piperazine-containing 1,2,4-triazole thione derivatives Chinese Chemical Letters. ,vol. 27, pp. 163- 167 ,(2016) , 10.1016/J.CCLET.2015.09.015

Klaus Stenzel, Ulrich Heinemann, Stefan Dutzmann, Fungicidal active substance combinations ,(1999)

Jan Rybniker, Anthony Vocat, Claudia Sala, Philippe Busso, Florence Pojer, Andrej Benjak, Stewart T. Cole, Lansoprazole is an antituberculous prodrug targeting cytochrome bc1. Nature Communications. ,vol. 6, pp. 7659- 7659 ,(2015) , 10.1038/NCOMMS8659