Synthesis and anticancer evaluation of imidazolinone and benzoxazole derivatives

作者: Heba A. El-Hady , Samar A. Abubshait

DOI: 10.1016/J.ARABJC.2014.05.006

关键词:

摘要: Abstract A series of imidazolinone and benzoxazole derivatives ( 3 5 ) have been synthesized by the condensation oxazolinone 2a – c with aniline 2-hydroxyaniline. Acetyl 4 , 6 7 were prepared via acetylation compounds acetic anhydride chloroacetyl chloride. The results revealed that are potent against cancer cell lines MCF-7 HePG2. In particular, more than derivatives.

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