Crystalline forms of a pyridine derivative
作者： David Clapham , Claire Louise Anderton , Ronnie Maxwell Lawrence
DOI:
关键词:
摘要: The invention relates to 4-methylbenzenesulfonate salt of the compound Formula (I) in a crystalline form or solvate thereof, pharmaceutical formulations containing them, their use therapy and processes for preparing same.
lens.org 参考文章(17)
Carl M. Mendel, Alteration of circadian rhythmicity with a tachykinin antagonist ,(1997)
Andreas Koblet, Jens-Uwe Peters, Patrick Schnider, Andrew Sleight, Heinz Stadler, Torsten Hoffmann, Dual nk1/nk3 receptor antagonists ,(2009)
Sandro Belvedere, Alessandro Falchi, Romano Di Fabio, Daniele Andreotti, Riccardo Giovannini, Giuseppe Alvaro, Pyridine derivatives and their use in the treatment of psychotic disorders ,(2006)
Andreas Koblet, Jens-Uwe Peters, Patrick Schnider, Andrew Sleight, Heinz Stadler, Torsten Hoffmann, Dual nk1/nk3 antagonists for treating schizophrenia ,(2004)
Heather Finlay, Yoon T Jeon, Serge Beaudoin, John Lloyd, Lin Yan, Michael Francis Gross, Heterocyclo inhibitors of potassium channel function ,(2003)
Angelo Gavezzotti, Are Crystal Structures Predictable Accounts of Chemical Research. ,vol. 27, pp. 309- 314 ,(1994) , 10.1021/AR00046A004
Etienne Challet, Christine Dugovic, Fred W. Turek, Olivier Van Reeth, The selective neurokinin 1 receptor antagonist R116301 modulates photic responses of the hamster circadian system. Neuropharmacology. ,vol. 40, pp. 408- 415 ,(2001) , 10.1016/S0028-3908(00)00165-9
Etienne Challet, Erik Naylor, Joseph M Metzger, D.Euan MacIntyre, Fred W Turek, An NK1 receptor antagonist affects the circadian regulation of locomotor activity in golden hamsters. Brain Research. ,vol. 800, pp. 32- 39 ,(1998) , 10.1016/S0006-8993(98)00491-0
Yoshinori IKEURA, Toshimasa TANAKA, Yutaka KIYOTA, Shinji MORIMOTO, Masaki OGINO, Takenori ISHIMARU, Izumi KAMO, Takayuki DOI, Hideaki NATSUGARI, Potent NK1 receptor antagonists: synthesis and antagonistic activity of various heterocycles with an N-[3,5-bis(trifluoromethyl)benzyl]-N-methylcarbamoyl substituent. Chemical & Pharmaceutical Bulletin. ,vol. 45, pp. 1642- 1652 ,(1997) , 10.1248/CPB.45.1642
R. Ciccocioppo, I. Panocka, P. Pompei, G. de Caro, M. Massi, Selective agonists at NK3 tachykinin receptors inhibit alcohol intake in Sardinian alcohol-preferring rats Brain Research Bulletin. ,vol. 33, pp. 71- 77 ,(1994) , 10.1016/0361-9230(94)90050-7